[1] |
鞠强. 中外痤疮指南药物治疗之亮点[J]. 中华皮肤科杂志, 2017,50(6):459⁃462. doi: 10.3760/cma.j.issn.0412⁃4030.2017. 06.024.
|
[2] |
Cong TX, Hao D, Wen X, et al. From pathogenesis of acne vulgaris to anti⁃acne agents[J]. Arch Dermatol Res, 2019,311(5):337⁃349. doi: 10.1007/s00403⁃019⁃01908⁃x.
|
[3] |
Zhanel G, Critchley I, Lin LY, et al. Microbiological profile of sarecycline, a novel targeted spectrum tetracycline for the treatment of acne vulgaris[J]. Antimicrob Agents Chemother, 2019,63(1):e01297⁃18. doi: 10.1128/AAC.01297⁃18.
|
[4] |
Moore A, Green LJ, Bruce S, et al. Once⁃daily oral sarecycline 1.5 mg/kg/day is effective for moderate to severe acne vulgaris: results from two identically designed, phase 3, randomized, double⁃blind clinical trials[J]. J Drugs Dermatol, 2018,17(9):987⁃996.
|
[5] |
Asadi A, Abdi M, Kouhsari E, et al. Minocycline, focus on mechanisms of resistance, antibacterial activity, and clinical effectiveness: back to the future[J]. J Glob Antimicrob Resist, 2020,22:161⁃174. doi: 10.1016/j.jgar.2020.01.022.
|
[6] |
Dosik J, Ellman H, Stuart I. Topical minocycline foam 4%: results of four phase 1 studies evaluating the potential for phototoxicity, photoallergy, sensitization, and cumulative irritation[J]. J Immunotoxicol, 2019,16(1):133⁃139. doi: 10. 1080/1547691X.2019.1610117.
|
[7] |
Gold LS, Dhawan S, Weiss J, et al. A novel topical minocycline foam for the treatment of moderate⁃to⁃severe acne vulgaris: results of 2 randomized, double⁃blind, phase 3 studies[J]. J Am Acad Dermatol, 2019,80(1):168⁃177. doi: 10.1016/j.jaad.2018. 08.020.
|
[8] |
Raoof TJ, Hooper D, Moore A, et al. Efficacy and safety of a novel topical minocycline foam for the treatment of moderate to severe acne vulgaris: a phase 3 study[J]. J Am Acad Dermatol, 2020,82(4):832⁃837. doi: 10.1016/j.jaad.2019.05.078.
|
[9] |
Yin S, Luo J, Qian A, et al. Retinoids activate the irritant receptor TRPV1 and produce sensory hypersensitivity[J]. J Clin Invest, 2013,123(9):3941⁃3951. doi: 10.1172/JCI66413.
|
[10] |
Aubert J, Piwnica D, Bertino B, et al. Nonclinical and human pharmacology of the potent and selective topical retinoic acid receptor⁃γ agonist trifarotene[J]. Br J Dermatol, 2018,179(2):442⁃456. doi: 10.1111/bjd.16719.
|
[11] |
Tan J, Thiboutot D, Popp G, et al. Randomized phase 3 evaluation of trifarotene 50 μg/g cream treatment of moderate facial and truncal acne[J]. J Am Acad Dermatol, 2019,80(6):1691⁃1699. doi: 10.1016/j.jaad.2019.02.044.
|
[12] |
Blume⁃Peytavi U, Fowler J, Kemény L, et al. Long⁃term safety and efficacy of trifarotene 50 μg/g cream, a first⁃in⁃class RAR⁃γ selective topical retinoid, in patients with moderate facial and truncal acne[J]. J Eur Acad Dermatol Venereol, 2020,34(1):166⁃173. doi: 10.1111/jdv.15794.
|
[13] |
Ju Q, Tao T, Hu T, et al. Sex hormones and acne[J]. Clin Dermatol, 2017,35(2):130⁃137. doi: 10.1016/j.clindermatol.2016. 10.004.
|
[14] |
Park JH, Bienenfeld A, Orlow SJ, et al. The use of hormonal antiandrogen therapy in female patients with acne: a 10⁃year retrospective Study[J]. Am J Clin Dermatol, 2018,19(3):449⁃455. doi: 10.1007/s40257⁃018⁃0349⁃6.
|
[15] |
Rosette C, Agan FJ, Mazzetti A, et al. Cortexolone 17α⁃propionate (clascoterone) is a novel androgen receptor antagonist that inhibits production of lipids and inflammatory cytokines from sebocytes in vitro[J]. J Drugs Dermatol, 2019,18(5):412⁃418.
|
[16] |
Hebert A, Thiboutot D, Stein Gold L, et al. Efficacy and safety of topical clascoterone cream, 1%, for treatment in patients with facial acne: two phase 3 randomized clinical trials[J]. JAMA Dermatol, 2020,156(6):621⁃630. doi: 10.1001/jamadermatol. 2020.0465.
|
[17] |
Eichenfield L, Hebert A, Gold LS, et al. Open⁃label, long⁃term extension study to evaluate the safety of clascoterone (CB⁃03⁃01) cream, 1% twice daily, in patients with acne vulgaris[J]. J Am Acad Dermatol, 2020,83(2):477⁃485. doi: 10.1016/j.jaad. 2020.04.087.
|
[18] |
Keating GM. Adapalene 0.1%/benzoyl peroxide 2.5% gel: a review of its use in the treatment of acne vulgaris in patients aged ≥ 12 years[J]. Am J Clin Dermatol, 2011,12(6):407⁃420. doi: 10.2165/11208170⁃000000000⁃00000.
|
[19] |
Seidler EM, Kimball AB. Meta⁃analysis comparing efficacy of benzoyl peroxide, clindamycin, benzoyl peroxide with salicylic acid, and combination benzoyl peroxide/clindamycin in acne[J]. J Am Acad Dermatol, 2010,63(1):52⁃62. doi: 10.1016/j.jaad.2009.07.052.
|
[20] |
Amar L, Kircik LH. Treatment of moderate acne vulgaris in fitzpatrick skin type Ⅴ or Ⅵ: efficacy and tolerability of fixed combination clindamycin phosphate 1.2%/benzoyl peroxide 3.75% gel[J]. J Drugs Dermatol, 2018,17(10):1107⁃1112.
|
[21] |
Zouboulis CC, Fischer TC, Wohlrab J, et al. Study of the efficacy, tolerability, and safety of 2 fixed⁃dose combination gels in the management of acne vulgaris[J]. Cutis, 2009,84(4):223⁃229.
|
[22] |
Weiss J, Stein Gold L, Leoni M, et al. Customized single⁃agent therapy management of severe inflammatory acne: a randomized, double⁃blind, parallel⁃group, controlled study of a new treatment⁃⁃adapalene 0.3%⁃benzoyl peroxide 2.5% gel[J]. J Drugs Dermatol, 2015,14(12):1427⁃1435.
|
[23] |
Gold MH, Baldwin H, Lin T. Management of comedonal acne vulgaris with fixed⁃combination topical therapy[J]. J Cosmet Dermatol, 2018,17(2):227⁃231. doi: 10.1111/jocd.12497.
|
[24] |
Ghaoui N, Hanna E, Abbas O, et al. Update on the use of dapsone in dermatology[J]. Int J Dermatol, 2020,59(7):787⁃795. doi: 10.1111/ijd.14761.
|
[25] |
Stein Gold LF, Jarratt MT, Bucko AD, et al. Efficacy and safety of once⁃daily dapsone gel, 7.5% for treatment of adolescents and adults with acne vulgaris: first of two identically designed, large, multicenter, randomized, vehicle⁃controlled trials[J]. J Drugs Dermatol, 2016,15(5):553⁃561.
|
[26] |
Eichenfield LF, Lain T, Frankel EH, et al. Efficacy and safety of once⁃daily dapsone gel, 7.5% for treatment of adolescents and adults with acne vulgaris: second of two identically designed, large, multicenter, randomized, vehicle⁃controlled trials[J]. J Drugs Dermatol, 2016,15(8):962⁃969.
|
[27] |
Jarratt MT, Jones TM, Chang⁃Lin JE, et al. Safety and pharmacokinetics of once⁃daily dapsone gel, 7.5% in Patients With Moderate Acne Vulgaris[J]. J Drugs Dermatol, 2016,15(10):1250⁃1259.
|
[28] |
Yale S, Stefanko N, McCarthy P, et al. Severe methemoglobinemia due to topical dapsone misuse in a teenage girl[J]. Pediatr Dermatol, 2020,37(2):377⁃378. doi: 10.1111/pde.14080.
|
[29] |
Jones ML, Ganopolsky JG, Labbé A, et al. Antimicrobial properties of nitric oxide and its application in antimicrobial formulations and medical devices[J]. Appl Microbiol Biotechnol, 2010,88(2):401⁃407. doi: 10.1007/s00253⁃010⁃2733⁃x.
|
[30] |
Qin M, Landriscina A, Rosen JM, et al. Nitric oxide⁃releasing nanoparticles prevent propionibacterium acnes⁃induced inflammation by both clearing the organism and inhibiting microbial stimulation of the innate immune response[J]. J Invest Dermatol, 2015,135(11):2723⁃2731. doi: 10.1038/jid. 2015.277.
|
[31] |
Hebert A,Del Rosso J, Rico M, et al.Evaluation of the efficacy, safety and tolerability of SB204 4% once⁃daily in subjects with moderate to severe acne vulgaris treated topically for up to 52 weeks [R/OL]//American Academy of Dermatology (AAD) Annual Meeting, San Diego, 2018[2020⁃06⁃01]. http: //novan.com/files/3115/1913/6178/SB204_Phase_3_AAD_Latebreaker_Presentation_vf.pdf.
|
[32] |
Melnik BC. Olumacostat glasaretil, a promising topical sebum⁃suppressing agent that affects all major pathogenic factors of acne vulgaris[J]. J Invest Dermatol, 2017,137(7):1405⁃1408. doi: 10.1016/j.jid.2017.01.026.
|
[33] |
Dermira, Inc. Dermira′s two phase 3 trials evaluating olumacostat glasaretil in patients with acne vulgaris did not meet co⁃ primary endpoints [EB/OL]. (2018⁃03⁃05)[2020⁃06⁃01]. https://investor.dermira.com/news⁃releases/press⁃release⁃details/2018/Dermiras⁃Two⁃Phase⁃3⁃Trials⁃Evaluating⁃Olumacostat⁃Glasaretil⁃in⁃Patients⁃with⁃Acne⁃Vulgaris⁃Did⁃Not⁃Meet⁃Co⁃Primary⁃Endpoints/default.aspx.
|
[34] |
Valente Duarte De Sousa IC. New and emerging drugs for the treatment of acne vulgaris in adolescents[J]. Expert Opin Pharmacother, 2019,20(8):1009⁃1024. doi: 10.1080/14656566. 2019.1584182.
|